                         SEQUENCE LISTING

<110>  biOasis Technologies, Inc.
 
<120>  CNS-TARGETED CONJUGATES HAVING MODIFIED FC REGIONS AND METHODS OF
        USE THEREOF

<130>  BIOA-007/01WO

<150>  US 61/870,914
<151>  2013-08-28

<160>  261   

<170>  PatentIn version 3.5

<210>  1
<211>  738
<212>  PRT
<213>  Homo sapiens

<400>  1

Met Arg Gly Pro Ser Gly Ala Leu Trp Leu Leu Leu Ala Leu Arg Thr 
1               5                   10                  15      


Val Leu Gly Gly Met Glu Val Arg Trp Cys Ala Thr Ser Asp Pro Glu 
            20                  25                  30          


Gln His Lys Cys Gly Asn Met Ser Glu Ala Phe Arg Glu Ala Gly Ile 
        35                  40                  45              


Gln Pro Ser Leu Leu Cys Val Arg Gly Thr Ser Ala Asp His Cys Val 
    50                  55                  60                  


Gln Leu Ile Ala Ala Gln Glu Ala Asp Ala Ile Thr Leu Asp Gly Gly 
65                  70                  75                  80  


Ala Ile Tyr Glu Ala Gly Lys Glu His Gly Leu Lys Pro Val Val Gly 
                85                  90                  95      


Glu Val Tyr Asp Gln Glu Val Gly Thr Ser Tyr Tyr Ala Val Ala Val 
            100                 105                 110         


Val Arg Arg Ser Ser His Val Thr Ile Asp Thr Leu Lys Gly Val Lys 
        115                 120                 125             


Ser Cys His Thr Gly Ile Asn Arg Thr Val Gly Trp Asn Val Pro Val 
    130                 135                 140                 


Gly Tyr Leu Val Glu Ser Gly Arg Leu Ser Val Met Gly Cys Asp Val 
145                 150                 155                 160 


Leu Lys Ala Val Ser Asp Tyr Phe Gly Gly Ser Cys Val Pro Gly Ala 
                165                 170                 175     


Gly Glu Thr Ser Tyr Ser Glu Ser Leu Cys Arg Leu Cys Arg Gly Asp 
            180                 185                 190         


Ser Ser Gly Glu Gly Val Cys Asp Lys Ser Pro Leu Glu Arg Tyr Tyr 
        195                 200                 205             


Asp Tyr Ser Gly Ala Phe Arg Cys Leu Ala Glu Gly Ala Gly Asp Val 
    210                 215                 220                 


Ala Phe Val Lys His Ser Thr Val Leu Glu Asn Thr Asp Gly Lys Thr 
225                 230                 235                 240 


Leu Pro Ser Trp Gly Gln Ala Leu Leu Ser Gln Asp Phe Glu Leu Leu 
                245                 250                 255     


Cys Arg Asp Gly Ser Arg Ala Asp Val Thr Glu Trp Arg Gln Cys His 
            260                 265                 270         


Leu Ala Arg Val Pro Ala His Ala Val Val Val Arg Ala Asp Thr Asp 
        275                 280                 285             


Gly Gly Leu Ile Phe Arg Leu Leu Asn Glu Gly Gln Arg Leu Phe Ser 
    290                 295                 300                 


His Glu Gly Ser Ser Phe Gln Met Phe Ser Ser Glu Ala Tyr Gly Gln 
305                 310                 315                 320 


Lys Asp Leu Leu Phe Lys Asp Ser Thr Ser Glu Leu Val Pro Ile Ala 
                325                 330                 335     


Thr Gln Thr Tyr Glu Ala Trp Leu Gly His Glu Tyr Leu His Ala Met 
            340                 345                 350         


Lys Gly Leu Leu Cys Asp Pro Asn Arg Leu Pro Pro Tyr Leu Arg Trp 
        355                 360                 365             


Cys Val Leu Ser Thr Pro Glu Ile Gln Lys Cys Gly Asp Met Ala Val 
    370                 375                 380                 


Ala Phe Arg Arg Gln Arg Leu Lys Pro Glu Ile Gln Cys Val Ser Ala 
385                 390                 395                 400 


Lys Ser Pro Gln His Cys Met Glu Arg Ile Gln Ala Glu Gln Val Asp 
                405                 410                 415     


Ala Val Thr Leu Ser Gly Glu Asp Ile Tyr Thr Ala Gly Lys Thr Tyr 
            420                 425                 430         


Gly Leu Val Pro Ala Ala Gly Glu His Tyr Ala Pro Glu Asp Ser Ser 
        435                 440                 445             


Asn Ser Tyr Tyr Val Val Ala Val Val Arg Arg Asp Ser Ser His Ala 
    450                 455                 460                 


Phe Thr Leu Asp Glu Leu Arg Gly Lys Arg Ser Cys His Ala Gly Phe 
465                 470                 475                 480 


Gly Ser Pro Ala Gly Trp Asp Val Pro Val Gly Ala Leu Ile Gln Arg 
                485                 490                 495     


Gly Phe Ile Arg Pro Lys Asp Cys Asp Val Leu Thr Ala Val Ser Glu 
            500                 505                 510         


Phe Phe Asn Ala Ser Cys Val Pro Val Asn Asn Pro Lys Asn Tyr Pro 
        515                 520                 525             


Ser Ser Leu Cys Ala Leu Cys Val Gly Asp Glu Gln Gly Arg Asn Lys 
    530                 535                 540                 


Cys Val Gly Asn Ser Gln Glu Arg Tyr Tyr Gly Tyr Arg Gly Ala Phe 
545                 550                 555                 560 


Arg Cys Leu Val Glu Asn Ala Gly Asp Val Ala Phe Val Arg His Thr 
                565                 570                 575     


Thr Val Phe Asp Asn Thr Asn Gly His Asn Ser Glu Pro Trp Ala Ala 
            580                 585                 590         


Glu Leu Arg Ser Glu Asp Tyr Glu Leu Leu Cys Pro Asn Gly Ala Arg 
        595                 600                 605             


Ala Glu Val Ser Gln Phe Ala Ala Cys Asn Leu Ala Gln Ile Pro Pro 
    610                 615                 620                 


His Ala Val Met Val Arg Pro Asp Thr Asn Ile Phe Thr Val Tyr Gly 
625                 630                 635                 640 


Leu Leu Asp Lys Ala Gln Asp Leu Phe Gly Asp Asp His Asn Lys Asn 
                645                 650                 655     


Gly Phe Lys Met Phe Asp Ser Ser Asn Tyr His Gly Gln Asp Leu Leu 
            660                 665                 670         


Phe Lys Asp Ala Thr Val Arg Ala Val Pro Val Gly Glu Lys Thr Thr 
        675                 680                 685             


Tyr Arg Gly Trp Leu Gly Leu Asp Tyr Val Ala Ala Leu Glu Gly Met 
    690                 695                 700                 


Ser Ser Gln Gln Cys Ser Gly Ala Ala Ala Pro Ala Pro Gly Ala Pro 
705                 710                 715                 720 


Leu Leu Pro Leu Leu Leu Pro Ala Leu Ala Ala Arg Leu Leu Pro Pro 
                725                 730                 735     


Ala Leu 
        


<210>  2
<211>  692
<212>  PRT
<213>  Homo sapiens

<400>  2

Gly Met Glu Val Arg Trp Cys Ala Thr Ser Asp Pro Glu Gln His Lys 
1               5                   10                  15      


Cys Gly Asn Met Ser Glu Ala Phe Arg Glu Ala Gly Ile Gln Pro Ser 
            20                  25                  30          


Leu Leu Cys Val Arg Gly Thr Ser Ala Asp His Cys Val Gln Leu Ile 
        35                  40                  45              


Ala Ala Gln Glu Ala Asp Ala Ile Thr Leu Asp Gly Gly Ala Ile Tyr 
    50                  55                  60                  


Glu Ala Gly Lys Glu His Gly Leu Lys Pro Val Val Gly Glu Val Tyr 
65                  70                  75                  80  


Asp Gln Glu Val Gly Thr Ser Tyr Tyr Ala Val Ala Val Val Arg Arg 
                85                  90                  95      


Ser Ser His Val Thr Ile Asp Thr Leu Lys Gly Val Lys Ser Cys His 
            100                 105                 110         


Thr Gly Ile Asn Arg Thr Val Gly Trp Asn Val Pro Val Gly Tyr Leu 
        115                 120                 125             


Val Glu Ser Gly Arg Leu Ser Val Met Gly Cys Asp Val Leu Lys Ala 
    130                 135                 140                 


Val Ser Asp Tyr Phe Gly Gly Ser Cys Val Pro Gly Ala Gly Glu Thr 
145                 150                 155                 160 


Ser Tyr Ser Glu Ser Leu Cys Arg Leu Cys Arg Gly Asp Ser Ser Gly 
                165                 170                 175     


Glu Gly Val Cys Asp Lys Ser Pro Leu Glu Arg Tyr Tyr Asp Tyr Ser 
            180                 185                 190         


Gly Ala Phe Arg Cys Leu Ala Glu Gly Ala Gly Asp Val Ala Phe Val 
        195                 200                 205             


Lys His Ser Thr Val Leu Glu Asn Thr Asp Gly Lys Thr Leu Pro Ser 
    210                 215                 220                 


Trp Gly Gln Ala Leu Leu Ser Gln Asp Phe Glu Leu Leu Cys Arg Asp 
225                 230                 235                 240 


Gly Ser Arg Ala Asp Val Thr Glu Trp Arg Gln Cys His Leu Ala Arg 
                245                 250                 255     


Val Pro Ala His Ala Val Val Val Arg Ala Asp Thr Asp Gly Gly Leu 
            260                 265                 270         


Ile Phe Arg Leu Leu Asn Glu Gly Gln Arg Leu Phe Ser His Glu Gly 
        275                 280                 285             


Ser Ser Phe Gln Met Phe Ser Ser Glu Ala Tyr Gly Gln Lys Asp Leu 
    290                 295                 300                 


Leu Phe Lys Asp Ser Thr Ser Glu Leu Val Pro Ile Ala Thr Gln Thr 
305                 310                 315                 320 


Tyr Glu Ala Trp Leu Gly His Glu Tyr Leu His Ala Met Lys Gly Leu 
                325                 330                 335     


Leu Cys Asp Pro Asn Arg Leu Pro Pro Tyr Leu Arg Trp Cys Val Leu 
            340                 345                 350         


Ser Thr Pro Glu Ile Gln Lys Cys Gly Asp Met Ala Val Ala Phe Arg 
        355                 360                 365             


Arg Gln Arg Leu Lys Pro Glu Ile Gln Cys Val Ser Ala Lys Ser Pro 
    370                 375                 380                 


Gln His Cys Met Glu Arg Ile Gln Ala Glu Gln Val Asp Ala Val Thr 
385                 390                 395                 400 


Leu Ser Gly Glu Asp Ile Tyr Thr Ala Gly Lys Thr Tyr Gly Leu Val 
                405                 410                 415     


Pro Ala Ala Gly Glu His Tyr Ala Pro Glu Asp Ser Ser Asn Ser Tyr 
            420                 425                 430         


Tyr Val Val Ala Val Val Arg Arg Asp Ser Ser His Ala Phe Thr Leu 
        435                 440                 445             


Asp Glu Leu Arg Gly Lys Arg Ser Cys His Ala Gly Phe Gly Ser Pro 
    450                 455                 460                 


Ala Gly Trp Asp Val Pro Val Gly Ala Leu Ile Gln Arg Gly Phe Ile 
465                 470                 475                 480 


Arg Pro Lys Asp Cys Asp Val Leu Thr Ala Val Ser Glu Phe Phe Asn 
                485                 490                 495     


Ala Ser Cys Val Pro Val Asn Asn Pro Lys Asn Tyr Pro Ser Ser Leu 
            500                 505                 510         


Cys Ala Leu Cys Val Gly Asp Glu Gln Gly Arg Asn Lys Cys Val Gly 
        515                 520                 525             


Asn Ser Gln Glu Arg Tyr Tyr Gly Tyr Arg Gly Ala Phe Arg Cys Leu 
    530                 535                 540                 


Val Glu Asn Ala Gly Asp Val Ala Phe Val Arg His Thr Thr Val Phe 
545                 550                 555                 560 


Asp Asn Thr Asn Gly His Asn Ser Glu Pro Trp Ala Ala Glu Leu Arg 
                565                 570                 575     


Ser Glu Asp Tyr Glu Leu Leu Cys Pro Asn Gly Ala Arg Ala Glu Val 
            580                 585                 590         


Ser Gln Phe Ala Ala Cys Asn Leu Ala Gln Ile Pro Pro His Ala Val 
        595                 600                 605             


Met Val Arg Pro Asp Thr Asn Ile Phe Thr Val Tyr Gly Leu Leu Asp 
    610                 615                 620                 


Lys Ala Gln Asp Leu Phe Gly Asp Asp His Asn Lys Asn Gly Phe Lys 
625                 630                 635                 640 


Met Phe Asp Ser Ser Asn Tyr His Gly Gln Asp Leu Leu Phe Lys Asp 
                645                 650                 655     


Ala Thr Val Arg Ala Val Pro Val Gly Glu Lys Thr Thr Tyr Arg Gly 
            660                 665                 670         


Trp Leu Gly Leu Asp Tyr Val Ala Ala Leu Glu Gly Met Ser Ser Gln 
        675                 680                 685             


Gln Cys Ser Gly 
    690         


<210>  3
<211>  11
<212>  PRT
<213>  Homo sapiens

<400>  3

Trp Cys Ala Thr Ser Asp Pro Glu Gln His Lys 
1               5                   10      


<210>  4
<211>  11
<212>  PRT
<213>  Homo sapiens

<400>  4

Arg Ser Ser His Val Thr Ile Asp Thr Leu Lys 
1               5                   10      


<210>  5
<211>  13
<212>  PRT
<213>  Homo sapiens

<400>  5

Ser Ser His Val Thr Ile Asp Thr Leu Lys Gly Val Lys 
1               5                   10              


<210>  6
<211>  14
<212>  PRT
<213>  Homo sapiens

<400>  6

Leu Cys Arg Gly Asp Ser Ser Gly Glu Gly Val Cys Asp Lys 
1               5                   10                  


<210>  7
<211>  16
<212>  PRT
<213>  Homo sapiens

<400>  7

Gly Asp Ser Ser Gly Glu Gly Val Cys Asp Lys Ser Pro Leu Glu Arg 
1               5                   10                  15      


<210>  8
<211>  9
<212>  PRT
<213>  Homo sapiens

<400>  8

Tyr Tyr Asp Tyr Ser Gly Ala Phe Arg 
1               5                   


<210>  9
<211>  7
<212>  PRT
<213>  Homo sapiens

<400>  9

Ala Asp Val Thr Glu Trp Arg 
1               5           


<210>  10
<211>  9
<212>  PRT
<213>  Homo sapiens

<400>  10

Val Pro Ala His Ala Val Val Val Arg 
1               5                   


<210>  11
<211>  10
<212>  PRT
<213>  Homo sapiens

<400>  11

Ala Asp Thr Asp Gly Gly Leu Ile Phe Arg 
1               5                   10  


<210>  12
<211>  9
<212>  PRT
<213>  Homo sapiens

<400>  12

Cys Gly Asp Met Ala Val Ala Phe Arg 
1               5                   


<210>  13
<211>  11
<212>  PRT
<213>  Homo sapiens

<400>  13

Leu Lys Pro Glu Ile Gln Cys Val Ser Ala Lys 
1               5                   10      


<210>  14
<211>  12
<212>  PRT
<213>  Homo sapiens

<400>  14

Asp Ser Ser His Ala Phe Thr Leu Asp Glu Leu Arg 
1               5                   10          


<210>  15
<211>  13
<212>  PRT
<213>  Homo sapiens

<400>  15

Ser Glu Asp Tyr Glu Leu Leu Cys Pro Asn Gly Ala Arg 
1               5                   10              


<210>  16
<211>  15
<212>  PRT
<213>  Homo sapiens

<400>  16

Ala Gln Asp Leu Phe Gly Asp Asp His Asn Lys Asn Gly Phe Lys 
1               5                   10                  15  


<210>  17
<211>  40
<212>  PRT
<213>  Homo sapiens

<400>  17

Phe Ser Ser Glu Ala Tyr Gly Gln Lys Asp Leu Leu Phe Lys Asp Ser 
1               5                   10                  15      


Thr Ser Glu Leu Val Pro Ile Ala Thr Gln Thr Tyr Glu Ala Trp Leu 
            20                  25                  30          


Gly His Glu Tyr Leu His Ala Met 
        35                  40  


<210>  18
<211>  221
<212>  PRT
<213>  Homo sapiens

<400>  18

Glu Arg Ile Gln Ala Glu Gln Val Asp Ala Val Thr Leu Ser Gly Glu 
1               5                   10                  15      


Asp Ile Tyr Thr Ala Gly Lys Thr Tyr Gly Leu Val Pro Ala Ala Gly 
            20                  25                  30          


Glu His Tyr Ala Pro Glu Asp Ser Ser Asn Ser Tyr Tyr Val Val Ala 
        35                  40                  45              


Val Val Arg Arg Asp Ser Ser His Ala Phe Thr Leu Asp Glu Leu Arg 
    50                  55                  60                  


Gly Lys Arg Ser Cys His Ala Gly Phe Gly Ser Pro Ala Gly Trp Asp 
65                  70                  75                  80  


Val Pro Val Gly Ala Leu Ile Gln Arg Gly Phe Ile Arg Pro Lys Asp 
                85                  90                  95      


Cys Asp Val Leu Thr Ala Val Ser Glu Phe Phe Asn Ala Ser Cys Val 
            100                 105                 110         


Pro Val Asn Asn Pro Lys Asn Tyr Pro Ser Ser Leu Cys Ala Leu Cys 
        115                 120                 125             


Val Gly Asp Glu Gln Gly Arg Asn Lys Cys Val Gly Asn Ser Gln Glu 
    130                 135                 140                 


Arg Tyr Tyr Gly Tyr Arg Gly Ala Phe Arg Cys Leu Val Glu Asn Ala 
145                 150                 155                 160 


Gly Asp Val Ala Phe Val Arg His Thr Thr Val Phe Asp Asn Thr Asn 
                165                 170                 175     


Gly His Asn Ser Glu Pro Trp Ala Ala Glu Leu Arg Ser Glu Asp Tyr 
            180                 185                 190         


Glu Leu Leu Cys Pro Asn Gly Ala Arg Ala Glu Val Ser Gln Phe Ala 
        195                 200                 205             


Ala Cys Asn Leu Ala Gln Ile Pro Pro His Ala Val Met 
    210                 215                 220     


<210>  19
<211>  32
<212>  PRT
<213>  Homo sapiens

<400>  19

Val Arg Pro Asp Thr Asn Ile Phe Thr Val Tyr Gly Leu Leu Asp Lys 
1               5                   10                  15      


Ala Gln Asp Leu Phe Gly Asp Asp His Asn Lys Asn Gly Phe Lys Met 
            20                  25                  30          


<210>  20
<211>  323
<212>  PRT
<213>  Homo sapiens

<400>  20

Tyr Ser Arg Glu Lys Asn Gln Pro Lys Pro Ser Pro Lys Arg Glu Ser 
1               5                   10                  15      


Gly Glu Glu Phe Arg Met Glu Lys Leu Asn Gln Leu Trp Glu Lys Ala 
            20                  25                  30          


Gln Arg Leu His Leu Pro Pro Val Arg Leu Ala Glu Leu His Ala Asp 
        35                  40                  45              


Leu Lys Ile Gln Glu Arg Asp Glu Leu Ala Trp Lys Lys Leu Lys Leu 
    50                  55                  60                  


Asp Gly Leu Asp Glu Asp Gly Glu Lys Glu Ala Arg Leu Ile Arg Asn 
65                  70                  75                  80  


Leu Asn Val Ile Leu Ala Lys Tyr Gly Leu Asp Gly Lys Lys Asp Ala 
                85                  90                  95      


Arg Gln Val Thr Ser Asn Ser Leu Ser Gly Thr Gln Glu Asp Gly Leu 
            100                 105                 110         


Asp Asp Pro Arg Leu Glu Lys Leu Trp His Lys Ala Lys Thr Ser Gly 
        115                 120                 125             


Lys Phe Ser Gly Glu Glu Leu Asp Lys Leu Trp Arg Glu Phe Leu His 
    130                 135                 140                 


His Lys Glu Lys Val His Glu Tyr Asn Val Leu Leu Glu Thr Leu Ser 
145                 150                 155                 160 


Arg Thr Glu Glu Ile His Glu Asn Val Ile Ser Pro Ser Asp Leu Ser 
                165                 170                 175     


Asp Ile Lys Gly Ser Val Leu His Ser Arg His Thr Glu Leu Lys Glu 
            180                 185                 190         


Lys Leu Arg Ser Ile Asn Gln Gly Leu Asp Arg Leu Arg Arg Val Ser 
        195                 200                 205             


His Gln Gly Tyr Ser Thr Glu Ala Glu Phe Glu Glu Pro Arg Val Ile 
    210                 215                 220                 


Asp Leu Trp Asp Leu Ala Gln Ser Ala Asn Leu Thr Asp Lys Glu Leu 
225                 230                 235                 240 


Glu Ala Phe Arg Glu Glu Leu Lys His Phe Glu Ala Lys Ile Glu Lys 
                245                 250                 255     


His Asn His Tyr Gln Lys Gln Leu Glu Ile Ala His Glu Lys Leu Arg 
            260                 265                 270         


His Ala Glu Ser Val Gly Asp Gly Glu Arg Val Ser Arg Ser Arg Glu 
        275                 280                 285             


Lys His Ala Leu Leu Glu Gly Arg Thr Lys Glu Leu Gly Tyr Thr Val 
    290                 295                 300                 


Lys Lys His Leu Gln Asp Leu Ser Gly Arg Ile Ser Arg Ala Arg His 
305                 310                 315                 320 


Asn Glu Leu 
            


<210>  21
<211>  58
<212>  PRT
<213>  Bos taurus

<400>  21

Arg Pro Asp Phe Cys Leu Glu Pro Pro Tyr Thr Gly Pro Cys Lys Ala 
1               5                   10                  15      


Arg Ile Ile Arg Tyr Phe Tyr Asn Ala Lys Ala Gly Leu Cys Gln Thr 
            20                  25                  30          


Phe Val Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Ser Ala 
        35                  40                  45              


Glu Asp Cys Met Arg Thr Cys Gly Gly Ala 
    50                  55              


<210>  22
<211>  19
<212>  PRT
<213>  Bos taurus

<400>  22

Thr Phe Val Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Ser 
1               5                   10                  15      


Ala Glu Asp 
            


<210>  23
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  23

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  24
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  24

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  25
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  25

Thr Phe Val Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Ser 
1               5                   10                  15      


Ala Glu Asp 
            


<210>  26
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  26

Thr Phe Gln Tyr Gly Gly Cys Met Gly Asn Gly Asn Asn Phe Val Thr 
1               5                   10                  15      


Glu Lys Glu 
            


<210>  27
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  27

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Asn Arg Asn Asn Phe Asp Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  28
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  28

Ser Phe Tyr Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Glu Glu Glu 
            


<210>  29
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  29

Thr Phe Phe Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  30
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  30

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  31
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  31

Thr Phe Phe Tyr Gly Gly Cys Arg Ala Lys Lys Asn Asn Tyr Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  32
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  32

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Lys Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  33
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  33

Thr Phe Gln Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  34
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  34

Thr Phe Gln Tyr Gly Gly Cys Arg Gly Lys Lys Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  35
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  35

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  36
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  36

Thr Phe Phe Tyr Gly Gly Ser Leu Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  37
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  37

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Lys Lys Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  38
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  38

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Gly Asn Asn Tyr Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  39
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  39

Pro Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Leu Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  40
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  40

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  41
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  41

Pro Phe Phe Tyr Gly Gly Cys Arg Ala Lys Lys Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Glu 
            


<210>  42
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  42

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Asp 
            


<210>  43
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  43

Thr Phe Phe Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Asp Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  44
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  44

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Lys Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  45
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  45

Pro Phe Phe Tyr Gly Gly Cys Gly Ala Asn Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  46
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  46

Thr Phe Phe Tyr Gly Gly Cys Gly Gly Lys Lys Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  47
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  47

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Arg Asn Asn Phe Leu Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  48
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  48

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  49
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  49

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Asn Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  50
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  50

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Gly Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  51
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  51

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Arg Asn Asn Phe Leu Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  52
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  52

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  53
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  53

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Gly Asn Asn Phe Lys Ser 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  54
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  54

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Lys Asn Asn Phe Asp Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  55
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  55

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Leu Arg 
1               5                   10                  15      


Glu Lys Glu 
            


<210>  56
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  56

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Gly Asn Asn Phe Asp Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  57
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  57

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Gly Asn Asn Phe Asp Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  58
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  58

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Gly Asn Asn Phe Val Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  59
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  59

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Lys Gly Asn Asn Tyr Val Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  60
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  60

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Lys Gly Asn Asn Phe Leu Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  61
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  61

Ser Phe Phe Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Phe Leu Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  62
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  62

Thr Phe Phe Tyr Gly Gly Cys Gly Gly Asn Lys Asn Asn Phe Val Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  63
<211>  12
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  63

Leu Gly Asn Lys Asn Asn Tyr Val Arg Glu Lys Tyr 
1               5                   10          


<210>  64
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  64

Thr Phe Phe Tyr Gly Gly Cys Gly Gly Asn Gly Asn Asn Phe Leu Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  65
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  65

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Arg Asn Asn Phe Leu Thr 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  66
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  66

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Gly Asn Asn Phe Lys Ser 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  67
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  67

Pro Phe Phe Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  68
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  68

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  69
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  69

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Asp 
            


<210>  70
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  70

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Asn Gly Asn Asn Phe Val Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  71
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  71

Ser Phe Phe Tyr Gly Gly Cys Met Gly Asn Gly Asn Asn Phe Val Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  72
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  72

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Asn Gly Asn Asn Phe Leu Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  73
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  73

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Gly Asn Asn Phe Val Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  74
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  74

Ser Phe Phe Tyr Gly Gly Cys Leu Gly Asn Gly Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  75
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  75

Thr Phe Phe Tyr Gly Gly Ser Leu Gly Asn Gly Asn Asn Phe Val Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  76
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  76

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Asn Gly Asn Asn Phe Val Thr 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  77
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  77

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Lys Gly Asn Asn Phe Val Ser 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  78
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  78

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Arg Asn Asn Phe Asp Arg 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  79
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  79

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Arg Asn Asn Phe Leu Arg 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  80
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  80

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  81
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  81

Pro Phe Phe Tyr Gly Gly Cys Gly Gly Asn Arg Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  82
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  82

Pro Phe Phe Tyr Gly Gly Ser Gly Gly Asn Arg Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  83
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  83

Met Arg Pro Asp Phe Cys Leu Glu Pro Pro Tyr Thr Gly Pro Cys Val 
1               5                   10                  15      


Ala Arg Ile 
            


<210>  84
<211>  21
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  84

Ala Arg Ile Ile Arg Tyr Phe Tyr Asn Ala Lys Ala Gly Leu Cys Gln 
1               5                   10                  15      


Thr Phe Val Tyr Gly 
            20      


<210>  85
<211>  22
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  85

Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Tyr Lys Ser Ala Glu Asp 
1               5                   10                  15      


Cys Met Arg Thr Cys Gly 
            20          


<210>  86
<211>  22
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  86

Pro Asp Phe Cys Leu Glu Pro Pro Tyr Thr Gly Pro Cys Val Ala Arg 
1               5                   10                  15      


Ile Ile Arg Tyr Phe Tyr 
            20          


<210>  87
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  87

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  88
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  88

Lys Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  89
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  89

Thr Phe Tyr Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Tyr Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  90
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  90

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  91
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  91

Cys Thr Phe Phe Tyr Gly Cys Cys Arg Gly Lys Arg Asn Asn Phe Lys 
1               5                   10                  15      


Thr Glu Glu Tyr 
            20  


<210>  92
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  92

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr Cys 
            20  


<210>  93
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  93

Thr Phe Phe Tyr Gly Gly Lys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  94
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  94

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Lys Arg Tyr 
            


<210>  95
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  95

Thr Phe Phe Tyr Gly Gly Lys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Glu Tyr 
            


<210>  96
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  96

Thr Phe Phe Tyr Gly Gly Lys Arg Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Gly Tyr 
            


<210>  97
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  97

Thr Phe Phe Tyr Gly Gly Lys Arg Gly Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Glu Lys Tyr 
            


<210>  98
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  98

Thr Phe Phe Tyr Gly Gly Lys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  99
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  99

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  100
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  100

Thr Phe Phe Tyr Gly Cys Gly Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  101
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  101

Thr Phe Phe Tyr Gly Gly Arg Cys Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  102
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  102

Thr Phe Phe Tyr Gly Gly Cys Leu Gly Asn Gly Asn Asn Phe Asp Thr 
1               5                   10                  15      


Glu Glu Glu Gln 
            20  


<210>  103
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  103

Thr Phe Gln Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  104
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  104

Tyr Asn Lys Glu Phe Gly Thr Phe Asn Thr Lys Gly Cys Glu Arg Gly 
1               5                   10                  15      


Tyr Arg Phe 
            


<210>  105
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  105

Arg Phe Lys Tyr Gly Gly Cys Leu Gly Asn Met Asn Asn Phe Glu Thr 
1               5                   10                  15      


Leu Glu Glu 
            


<210>  106
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  106

Arg Phe Lys Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Phe Leu Arg 
1               5                   10                  15      


Leu Lys Tyr 
            


<210>  107
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  107

Arg Phe Lys Tyr Gly Gly Cys Leu Gly Asn Lys Asn Asn Tyr Leu Arg 
1               5                   10                  15      


Leu Lys Tyr 
            


<210>  108
<211>  22
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  108

Lys Thr Lys Arg Lys Arg Lys Lys Gln Arg Val Lys Ile Ala Tyr Glu 
1               5                   10                  15      


Glu Ile Phe Lys Asn Tyr 
            20          


<210>  109
<211>  15
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  109

Lys Thr Lys Arg Lys Arg Lys Lys Gln Arg Val Lys Ile Ala Tyr 
1               5                   10                  15  


<210>  110
<211>  17
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  110

Arg Gly Gly Arg Leu Ser Tyr Ser Arg Arg Phe Ser Thr Ser Thr Gly 
1               5                   10                  15      


Arg 
    


<210>  111
<211>  10
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  111

Arg Arg Leu Ser Tyr Ser Arg Arg Arg Phe 
1               5                   10  


<210>  112
<211>  16
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  112

Arg Gln Ile Lys Ile Trp Phe Gln Asn Arg Arg Met Lys Trp Lys Lys 
1               5                   10                  15      


<210>  113
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  113

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  114
<211>  59
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  114

Met Arg Pro Asp Phe Cys Leu Glu Pro Pro Tyr Thr Gly Pro Cys Val 
1               5                   10                  15      


Ala Arg Ile Ile Arg Tyr Phe Tyr Asn Ala Lys Ala Gly Leu Cys Gln 
            20                  25                  30          


Thr Phe Val Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Ser 
        35                  40                  45              


Ala Glu Asp Cys Met Arg Thr Cys Gly Gly Ala 
    50                  55                  


<210>  115
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  115

Thr Phe Phe Tyr Gly Gly Cys Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Lys Glu Tyr 
            


<210>  116
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  116

Thr Phe Phe Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Arg 
1               5                   10                  15      


Ala Lys Tyr 
            


<210>  117
<211>  35
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  117

Asn Ala Lys Ala Gly Leu Cys Gln Thr Phe Val Tyr Gly Gly Cys Leu 
1               5                   10                  15      


Ala Lys Arg Asn Asn Phe Glu Ser Ala Glu Asp Cys Met Arg Thr Cys 
            20                  25                  30          


Gly Gly Ala 
        35  


<210>  118
<211>  24
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  118

Tyr Gly Gly Cys Arg Ala Lys Arg Asn Asn Phe Lys Ser Ala Glu Asp 
1               5                   10                  15      


Cys Met Arg Thr Cys Gly Gly Ala 
            20                  


<210>  119
<211>  22
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  119

Gly Leu Cys Gln Thr Phe Val Tyr Gly Gly Cys Arg Ala Lys Arg Asn 
1               5                   10                  15      


Asn Phe Lys Ser Ala Glu 
            20          


<210>  120
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  120

Leu Cys Gln Thr Phe Val Tyr Gly Gly Cys Glu Ala Lys Arg Asn Asn 
1               5                   10                  15      


Phe Lys Ser Ala 
            20  


<210>  121
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  121

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  122
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  122

Arg Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  123
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  123

Arg Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  124
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  124

Arg Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Arg Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  125
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  125

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Arg Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  126
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  126

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Arg Arg Asn Asn Phe Arg Thr 
1               5                   10                  15      


Glu Glu Tyr 
            


<210>  127
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  127

Cys Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys 
1               5                   10                  15      


Thr Glu Glu Tyr 
            20  


<210>  128
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  128

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Lys Arg Asn Asn Phe Lys Thr 
1               5                   10                  15      


Glu Glu Tyr Cys 
            20  


<210>  129
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  129

Cys Thr Phe Phe Tyr Gly Gly Ser Arg Gly Arg Arg Asn Asn Phe Arg 
1               5                   10                  15      


Thr Glu Glu Tyr 
            20  


<210>  130
<211>  20
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Aprotinin analogue peptide

<400>  130

Thr Phe Phe Tyr Gly Gly Ser Arg Gly Arg Arg Asn Asn Phe Arg Thr 
1               5                   10                  15      


Glu Glu Tyr Cys 
            20  


<210>  131
<211>  86
<212>  PRT
<213>  Human immunodeficiency virus-1

<400>  131

Met Glu Pro Val Asp Pro Arg Leu Glu Pro Trp Lys His Pro Gly Ser 
1               5                   10                  15      


Gln Pro Lys Thr Ala Cys Thr Thr Cys Tyr Cys Lys Lys Cys Cys Phe 
            20                  25                  30          


His Cys Gln Val Cys Phe Thr Thr Lys Ala Leu Gly Ile Ser Tyr Gly 
        35                  40                  45              


Arg Lys Lys Arg Arg Gln Arg Arg Arg Pro Pro Gln Gly Ser Gln Thr 
    50                  55                  60                  


His Gln Val Ser Leu Ser Lys Gln Pro Thr Ser Gln Pro Arg Gly Asp 
65                  70                  75                  80  


Pro Thr Gly Pro Lys Glu 
                85      


<210>  132
<211>  20
<212>  PRT
<213>  Human immunodeficiency virus-1

<400>  132

Phe Thr Thr Lys Ala Leu Gly Ile Ser Tyr Gly Arg Lys Lys Arg Arg 
1               5                   10                  15      


Gln Arg Arg Arg 
            20  


<210>  133
<211>  16
<212>  PRT
<213>  Drosiphila melanogaster

<400>  133

Arg Gln Ile Lys Ile Trp Phe Gln Asn Arg Arg Met Lys Trp Lys Lys 
1               5                   10                  15      


<210>  134
<211>  18
<212>  PRT
<213>  Sus scrofa

<400>  134

Arg Gly Gly Arg Leu Cys Tyr Cys Arg Arg Arg Phe Cys Val Cys Val 
1               5                   10                  15      


Gly Arg 
        


<210>  135
<211>  19
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  PG-1 analogue peptide (SynB1)

<400>  135

Arg Gly Gly Arg Leu Ser Tyr Ser Arg Arg Arg Phe Ser Thr Ser Thr 
1               5                   10                  15      


Gly Arg Ala 
            


<210>  136
<211>  10
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  PG-1 analogue peptide (SynB3)

<400>  136

Arg Arg Leu Ser Tyr Ser Arg Arg Arg Phe 
1               5                   10  


<210>  137
<211>  17
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  PG-1 analogue peptide (SynB5)

<400>  137

Arg Gly Gly Arg Leu Ala Tyr Leu Arg Arg Arg Trp Ala Val Leu Gly 
1               5                   10                  15      


Arg 
    


<210>  138
<211>  12
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  138

His Leu Asp Cys Met Pro Arg Gly Cys Phe Arg Asn 
1               5                   10          


<210>  139
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  139

Ala Cys Gln Val Lys Ser Met Pro Arg Cys 
1               5                   10  


<210>  140
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  140

Ala Cys Thr Thr Pro Met Pro Arg Leu Cys 
1               5                   10  


<210>  141
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  141

Ala Cys Lys Ala Pro Gln Met Pro Arg Cys 
1               5                   10  


<210>  142
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  142

Ala Cys Leu Asn Pro Ser Met Pro Arg Cys 
1               5                   10  


<210>  143
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  143

Ala Cys Leu Val Ser Ser Met Pro Arg Cys 
1               5                   10  


<210>  144
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  144

Ala Cys Leu Gln Pro Met Pro Arg Leu Cys 
1               5                   10  


<210>  145
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  145

Ala Cys Pro Val Ser Ser Met Pro Arg Cys 
1               5                   10  


<210>  146
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  146

Ala Cys Gln Ser Pro Met Pro Arg Leu Cys 
1               5                   10  


<210>  147
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  147

Ala Cys Leu Thr Pro Met Pro Arg Leu Cys 
1               5                   10  


<210>  148
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  148

Asp Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  149
<211>  10
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  149

Ala Cys Met Pro Arg Leu Arg Gly Cys Ala 
1               5                   10  


<210>  150
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  150

Ala Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  151
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  151

Asp Ala Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  152
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  152

Asp Ser Ala Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  153
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  153

Asp Ser Gly Ala Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  154
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  154

Asp Ser Gly Leu Cys Met Pro Arg Ala Arg Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  155
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  155

Asp Ser Gly Leu Cys Met Pro Arg Leu Ala Gly Cys Asp Pro Arg 
1               5                   10                  15  


<210>  156
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  156

Asp Ser Gly Leu Cys Met Pro Arg Leu Arg Ala Cys Asp Pro Arg 
1               5                   10                  15  


<210>  157
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  157

Asp Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Ala Pro Arg 
1               5                   10                  15  


<210>  158
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  158

Asp Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Ala Arg 
1               5                   10                  15  


<210>  159
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  159

Asp Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Ala 
1               5                   10                  15  


<210>  160
<211>  14
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  160

Ser Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10                  


<210>  161
<211>  13
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  161

Gly Leu Cys Met Pro Arg Leu Arg Gly Cys Asp Pro Arg 
1               5                   10              


<210>  162
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  162

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  163
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  163

Cys Met Pro Arg Ala Arg Gly Cys 
1               5               


<210>  164
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  164

Cys Met Pro Arg Leu Ala Gly Cys 
1               5               


<210>  165
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  165

Cys Met Pro Arg Leu Arg Ala Cys 
1               5               


<210>  166
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  166

Cys Met Pro Arg Leu Lys Gly Cys 
1               5               


<210>  167
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<400>  167

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  168
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (5)..(5)
<223>  D-Leucine

<400>  168

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  169
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (6)..(6)
<223>  D-Arginine

<400>  169

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  170
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  D-Cysteine

<400>  170

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  171
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  D-Cysteine

<400>  171

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  172
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Xaa = Sarcosine (Sar)

<400>  172

Cys Met Pro Arg Leu Arg Xaa Cys 
1               5               


<210>  173
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  (D)-Cysteine

<400>  173

Cys Met Pro Arg Lys Arg Gly Cys 
1               5               


<210>  174
<211>  7
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  (D)-Cysteine

<400>  174

Cys Met Pro Arg Leu Arg Cys 
1               5           


<210>  175
<211>  7
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  (D)-Cysteine

<400>  175

Cys Met Pro Arg Leu Cys Arg 
1               5           


<210>  176
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  (D)-Cysteine

<400>  176

Cys Met Pro Arg Cys Leu Arg Gly 
1               5               


<210>  177
<211>  6
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  177

Cys Met Pro Arg Gly Cys 
1               5       


<210>  178
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = Penicillamine (Pen)

<400>  178

Xaa Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  179
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = D-Penicillamine (D-Pen)

<400>  179

Xaa Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  180
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  180

Cys Met Pro Arg Leu Arg Gly Xaa 
1               5               


<210>  181
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = Penicillamine (Pen)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  181

Xaa Met Pro Arg Leu Arg Gly Xaa 
1               5               


<210>  182
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = D-Penicillamine (D-Pen)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  182

Xaa Met Pro Arg Leu Arg Gly Xaa 
1               5               


<210>  183
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = D-Penicillamine (D-Pen)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = D-Penicillamine (D-Pen)

<400>  183

Xaa Met Pro Arg Leu Arg Gly Xaa 
1               5               


<210>  184
<211>  8
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = 3-Mercaptopropionic acid (Mpa)

<400>  184

Xaa Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  185
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  185

Met Thr Val Met Pro Thr Gly Leu Trp Asn Pro Leu Ile Pro Ser 
1               5                   10                  15  


<210>  186
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  186

Ser Ala Ser Trp Phe Ala Val Pro Ile Pro Pro Leu Arg Leu Glu 
1               5                   10                  15  


<210>  187
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  187

Met Thr Pro Met Ser Thr Pro Arg Met Leu Pro Val Tyr Val Ala 
1               5                   10                  15  


<210>  188
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  188

Met Thr Ala Thr His Leu Ser Thr Leu Phe Gln Pro Leu Thr Tyr 
1               5                   10                  15  


<210>  189
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  189

Met Ser Pro Ile Pro Pro Ala Ala Ser Thr Trp Ala Asn Thr Leu 
1               5                   10                  15  


<210>  190
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  190

Met Thr Ala Asn Pro Leu Gln Asn Ala Pro Gly Pro Leu Ser Leu 
1               5                   10                  15  


<210>  191
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  191

Met Gln Thr Ala Pro Pro Pro Pro Leu Thr Arg Val Gln Trp Ser 
1               5                   10                  15  


<210>  192
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  192

Gly Thr Pro Arg Met His Ile Pro Leu Asn Val Asp His Leu Pro 
1               5                   10                  15  


<210>  193
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  193

Leu Thr Leu Pro Pro Ile Ser Gly Leu Ser Ser Tyr Pro Leu Pro 
1               5                   10                  15  


<210>  194
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  194

Thr Pro Ser Ala His Ala Met Ala Leu Gln Ser Leu Ser Val Gly 
1               5                   10                  15  


<210>  195
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  195

Leu Thr Leu Pro Pro Ile Ser Gly Leu Ser Ser Tyr Pro Leu Pro 
1               5                   10                  15  


<210>  196
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  196

Met Gly Thr Leu Asn Ala Pro Thr Ala Tyr Pro Gln Asp Ser Leu 
1               5                   10                  15  


<210>  197
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  197

Leu Thr Asn Pro Pro Ala Tyr Leu Pro Gln Asn Thr Asp Pro His 
1               5                   10                  15  


<210>  198
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  198

Met Gly Leu Pro Leu Pro Tyr Ile Gln Thr Ile Leu His Thr Pro 
1               5                   10                  15  


<210>  199
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  199

Ser Ala Ala Leu Ile Ala Met Ser Ser Phe Lys Ser Ile Thr Ala 
1               5                   10                  15  


<210>  200
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  200

Ser Gly Phe Ala Phe Ala Arg Ser Val Pro Thr Glu Ser Arg Arg 
1               5                   10                  15  


<210>  201
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  201

Met Thr Ser Pro Tyr Met Ser Leu Pro Pro Ser Thr Asp Asp Met 
1               5                   10                  15  


<210>  202
<211>  15
<212>  PRT
<213>  artificial sequence

<220>
<223>  synthesized peptide

<400>  202

Leu Thr Asn Pro Pro Ala Tyr Leu Pro Gln Asn Thr Asp Pro His 
1               5                   10                  15  


<210>  203
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  hLDLR binding peptide motif


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Cysteine or an analogue or isostere thereof

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Proline or an analogue or isostere thereof

<220>
<221>  MOD_RES
<222>  (6)..(6)
<223>  Xaa = Ala or Arg

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Glycine or an analogue or isostere thereof

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Cysteine or an analogue or isostere thereof

<400>  203

Xaa Met Xaa Arg Leu Xaa Xaa Xaa 
1               5               


<210>  204
<211>  8
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  hLDLR binding peptide motif


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = Cys, D-Cys, Penicillamine (Pen) or D-Penicillamine (D-Pen)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pro, Pipecolic acid (Pip) or Thiazolidine-4-carboxylic acid
       (Thz)

<400>  204

Xaa Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  205
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<400>  205

Cys Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  206
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = D-Penicillamine (D-Pen)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<400>  206

Xaa Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  207
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = Penicillamine (Pen)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<400>  207

Xaa Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  208
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<400>  208

Cys Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  209
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = D-Penicillamine (D-Pen)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<400>  209

Xaa Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  210
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  Xaa = Penicillamine (Pen)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<400>  210

Xaa Met Xaa Arg Leu Arg Gly Cys 
1               5               


<210>  211
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine)

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Xaa = Sarcosine (Sar)

<400>  211

Cys Met Xaa Arg Leu Arg Xaa Cys 
1               5               


<210>  212
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  212

Cys Met Xaa Arg Leu Arg Gly Xaa 
1               5               


<210>  213
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Thiazolidine-4-carboxylic acid (Thz)

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Xaa = Sarcosine (Sar)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  213

Cys Met Xaa Arg Leu Arg Xaa Xaa 
1               5               


<210>  214
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Xaa = Sarcosine (Sar)

<400>  214

Cys Met Xaa Arg Leu Arg Xaa Cys 
1               5               


<210>  215
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  215

Cys Met Xaa Arg Leu Arg Gly Xaa 
1               5               


<210>  216
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (3)..(3)
<223>  Xaa = Pipecolic acid (Pip)

<220>
<221>  MOD_RES
<222>  (7)..(7)
<223>  Xaa = Sarcosine (Sar)

<220>
<221>  MOD_RES
<222>  (8)..(8)
<223>  Xaa = Penicillamine (Pen)

<400>  216

Cys Met Xaa Arg Leu Arg Xaa Xaa 
1               5               


<210>  217
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (4)..(4)
<223>  Xaa = hArg

<400>  217

Cys Met Pro Xaa Leu Arg Gly Cys 
1               5               


<210>  218
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (4)..(4)
<223>  Xaa = 2-amino-4-(N'-Pbf-guanidino)-butyric acid (Agb)

<400>  218

Cys Met Pro Xaa Leu Arg Gly Cys 
1               5               


<210>  219
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (4)..(4)
<223>  Xaa = 2-amino-4-(N'-Pbf-guanidino)-propanoic acid (Agp)

<400>  219

Cys Met Pro Xaa Leu Arg Gly Cys 
1               5               


<210>  220
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (4)..(4)
<223>  Xaa = Citrulline (Cit)

<400>  220

Cys Met Pro Xaa Leu Arg Gly Cys 
1               5               


<210>  221
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (6)..(6)
<223>  Xaa = Citrulline (Cit)

<400>  221

Cys Met Pro Arg Leu Xaa Gly Cys 
1               5               


<210>  222
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<220>
<221>  MOD_RES
<222>  (6)..(6)
<223>  Xaa = Arg(NO2)

<400>  222

Cys Met Pro Arg Leu Xaa Gly Cys 
1               5               


<210>  223
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized


<220>
<221>  MOD_RES
<222>  (1)..(1)
<223>  D-Cysteine

<400>  223

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  224
<211>  8
<212>  PRT
<213>  Artificial sequence

<220>
<223>  synthesized

<400>  224

Cys Met Pro Arg Leu Arg Gly Cys 
1               5               


<210>  225
<211>  230
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Synthetic Fc Construct


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  Xaa is Ala or absent

<220>
<221>  MISC_FEATURE
<222>  (16)..(16)
<223>  Xaa is Pro or Glu

<220>
<221>  MISC_FEATURE
<222>  (17)..(17)
<223>  Xaa is Phe, Val or Ala

<220>
<221>  MISC_FEATURE
<222>  (18)..(18)
<223>  Xaa is Leu, Glu or Ala

<220>
<221>  MISC_FEATURE
<222>  (80)..(80)
<223>  Xaa is Asn or Ala

<220>
<221>  MISC_FEATURE
<222>  (230)..(230)
<223>  Xaa is Lys or absent

<400>  225

Xaa Glu Ser Lys Tyr Gly Pro Pro Cys Pro Pro Cys Pro Ala Pro Xaa 
1               5                   10                  15      


Xaa Xaa Gly Gly Pro Ser Val Phe Leu Phe Pro Pro Lys Pro Lys Asp 
            20                  25                  30          


Thr Leu Met Ile Ser Arg Thr Pro Glu Val Thr Cys Val Val Val Asp 
        35                  40                  45              


Val Ser Gln Glu Asp Pro Glu Val Gln Phe Asn Trp Tyr Val Asp Gly 
    50                  55                  60                  


Val Glu Val His Asn Ala Lys Thr Lys Pro Arg Glu Glu Gln Phe Xaa 
65                  70                  75                  80  


Ser Thr Tyr Arg Val Val Ser Val Leu Thr Val Leu His Gln Asp Trp 
                85                  90                  95      


Leu Asn Gly Lys Glu Tyr Lys Cys Lys Val Ser Asn Lys Gly Leu Pro 
            100                 105                 110         


Ser Ser Ile Glu Lys Thr Ile Ser Lys Ala Lys Gly Gln Pro Arg Glu 
        115                 120                 125             


Pro Gln Val Tyr Thr Leu Pro Pro Ser Gln Glu Glu Met Thr Lys Asn 
    130                 135                 140                 


Gln Val Ser Leu Thr Cys Leu Val Lys Gly Phe Tyr Pro Ser Asp Ile 
145                 150                 155                 160 


Ala Val Glu Trp Glu Ser Asn Gly Gln Pro Glu Asn Asn Tyr Lys Thr 
                165                 170                 175     


Thr Pro Pro Val Leu Asp Ser Asp Gly Ser Phe Phe Leu Tyr Ser Arg 
            180                 185                 190         


Leu Thr Val Asp Lys Ser Arg Trp Gln Glu Gly Asn Val Phe Ser Cys 
        195                 200                 205             


Ser Val Met His Glu Ala Leu His Asn His Tyr Thr Gln Lys Ser Leu 
    210                 215                 220                 


Ser Leu Ser Leu Gly Xaa 
225                 230 


<210>  226
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sulfatase motif


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  Xaa = Any amino acid or absent

<220>
<221>  MISC_FEATURE
<222>  (2)..(2)
<223>  Xaa = Cys or Ser

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  Xaa = Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  Xaa = Pro or Ala

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  Xaa = Any amino acid

<400>  226

Xaa Xaa Xaa Xaa Xaa 
1               5   


<210>  227
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Sulfatase motifs


<220>
<221>  MISC_FEATURE
<222>  (1)..(1)
<223>  Xaa = Any amino acid or absent

<220>
<221>  MOD_RES
<222>  (2)..(2)
<223>  Formylglycine

<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  Xaa = Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (4)..(4)
<223>  Xaa = Pro or Ala

<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  Xaa = Any amino acid

<400>  227

Xaa Gly Xaa Xaa Xaa 
1               5   


<210>  228
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Ser linker

<400>  228

Gly Ser Gly Ser 
1               


<210>  229
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Ser linker

<400>  229

Gly Gly Ser Gly 
1               


<210>  230
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Ser linker

<400>  230

Gly Gly Gly Ser 
1               


<210>  231
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Ser linker

<400>  231

Gly Gly Gly Gly Ser 
1               5   


<210>  232
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Asn linker

<400>  232

Gly Asn Gly Asn 
1               


<210>  233
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Asn linker

<400>  233

Gly Gly Asn Gly 
1               


<210>  234
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Asn linker

<400>  234

Gly Gly Gly Asn 
1               


<210>  235
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Exemplary Gly Asn linker

<400>  235

Gly Gly Gly Gly Asn 
1               5   


<210>  236
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - thrombin cleavable

<400>  236

Gly Arg Gly Asp 
1               


<210>  237
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - thrombin cleavable

<400>  237

Gly Arg Gly Asp Asn Pro 
1               5       


<210>  238
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - thrombin cleavable

<400>  238

Gly Arg Gly Asp Ser 
1               5   


<210>  239
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - thrombin cleavable

<400>  239

Gly Arg Gly Asp Ser Pro Lys 
1               5           


<210>  240
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - elastase cleavable

<400>  240

Ala Ala Pro Val 
1               


<210>  241
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - elastase cleavable

<400>  241

Ala Ala Pro Leu 
1               


<210>  242
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - elastase cleavable

<400>  242

Ala Ala Pro Phe 
1               


<210>  243
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - elastase cleavable

<400>  243

Ala Ala Pro Ala 
1               


<210>  244
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - elastase cleavable

<400>  244

Ala Tyr Leu Val 
1               


<210>  245
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - matrix metalloproteinase 
       cleavable


<220>
<221>  MISC_FEATURE
<222>  (3)..(3)
<223>  Xaa = Any amino acid

<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  Xaa = Any amino acid

<400>  245

Gly Pro Xaa Gly Pro Xaa 
1               5       


<210>  246
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - matrix metalloproteinase 
       cleavable


<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  Xaa = Any amino acid

<400>  246

Gly Pro Leu Gly Pro Xaa 
1               5       


<210>  247
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - matrix metalloproteinase 
       cleavable


<220>
<221>  MISC_FEATURE
<222>  (6)..(6)
<223>  Xaa = Any amino acid

<400>  247

Gly Pro Ile Gly Pro Xaa 
1               5       


<210>  248
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - matrix metalloproteinase 
       cleavable


<220>
<221>  MISC_FEATURE
<222>  (5)..(5)
<223>  Xaa = Any amino acid

<400>  248

Ala Pro Gly Leu Xaa 
1               5   


<210>  249
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable


<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  Xaa = Any amino acid

<400>  249

Pro Leu Gly Pro Asp Arg Xaa 
1               5           


<210>  250
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable


<220>
<221>  MISC_FEATURE
<222>  (7)..(7)
<223>  Xaa = Any amino acid

<400>  250

Pro Leu Gly Leu Leu Gly Xaa 
1               5           


<210>  251
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable

<400>  251

Pro Gln Gly Ile Ala Gly Trp 
1               5           


<210>  252
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable

<400>  252

Pro Leu Gly Cys His 
1               5   


<210>  253
<211>  6
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable

<400>  253

Pro Leu Gly Leu Tyr Ala 
1               5       


<210>  254
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable

<400>  254

Pro Leu Ala Leu Trp Ala Arg 
1               5           


<210>  255
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - collagenase cleavable

<400>  255

Pro Leu Ala Tyr Trp Ala Arg 
1               5           


<210>  256
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - stromelysin cleavable

<400>  256

Pro Tyr Ala Tyr Tyr Met Arg 
1               5           


<210>  257
<211>  7
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - gelatinase cleavable

<400>  257

Pro Leu Gly Met Tyr Ser Arg 
1               5           


<210>  258
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - angiotensin converting enzyme 
       cleavable

<400>  258

Gly Asp Lys Pro 
1               


<210>  259
<211>  5
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - angiotensin converting enzyme 
       cleavable

<400>  259

Gly Ser Asp Lys Pro 
1               5   


<210>  260
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - cathepsin B cleavable

<400>  260

Ala Leu Ala Leu 
1               


<210>  261
<211>  4
<212>  PRT
<213>  Artificial Sequence

<220>
<223>  Enzymatically degradable linker - cathepsin B cleavable

<400>  261

Gly Phe Leu Gly 
1               


