                         SEQUENCE LISTING

<110>  Beth Israel Deaconess Medical Center, Inc.
       LU, Kun Ping
       ZHOU, Xiao Zhen
       WEI, Shuo
 
<120>  ENHANCED ATRA-RELATED COMPOUNDS DERIVED FROM STRUCTURE-ACTIVITY 
       RELATIONSHIPS AND MODELING FOR INHIBITING PIN1

<130>  01948-239WO6

<150>  61/968,862
<151>  2014-03-21

<150>  Not Yet Assigned
<151>  2015-03-12

<160>  48    

<170>  PatentIn version 3.5

<210>  1
<211>  119
<212>  PRT
<213>  Homo sapiens

<400>  1

Gly Lys Asn Gly Gln Gly Glu Pro Ala Arg Val Arg Cys Ser His Leu 
1               5                   10                  15      


Leu Val Lys His Ser Gln Ser Arg Arg Pro Ser Ser Trp Arg Gln Glu 
            20                  25                  30          


Lys Ile Thr Arg Thr Lys Glu Glu Ala Leu Glu Leu Ile Asn Gly Tyr 
        35                  40                  45              


Ile Gln Lys Ile Lys Ser Gly Glu Glu Asp Phe Glu Ser Leu Ala Ser 
    50                  55                  60                  


Gln Phe Ser Asp Cys Ser Ser Ala Lys Ala Arg Gly Asp Leu Gly Ala 
65                  70                  75                  80  


Phe Ser Arg Gly Gln Met Gln Lys Pro Phe Glu Asp Ala Ser Phe Ala 
                85                  90                  95      


Leu Arg Thr Gly Glu Met Ser Gly Pro Val Phe Thr Asp Ser Gly Ile 
            100                 105                 110         


His Ile Ile Leu Arg Thr Glu 
        115                 


<210>  2
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  2
ccaccgtcac acagtattta t                                                 21


<210>  3
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  3
gctcgaatga taactattga t                                                 21


<210>  4
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  4
ccagtgcatg accttactat t                                                 21


<210>  5
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  5
catgagaagt atgacaacag cct                                               23


<210>  6
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  6
agtccttcca cgataccaaa gt                                                22


<210>  7
<211>  19
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  7
gcctcacagt tcagcgact                                                    19


<210>  8
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  8
actcagtgcg gaggatgatg t                                                 21


<210>  9
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  9
tgcccagaaa atgaaaaagg                                                   20


<210>  10
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  10
gtgtatgtgg caatgcgttc                                                   20


<210>  11
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  11
acagtggcca cctacaaagg                                                   20


<210>  12
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  12
ccgagatggg gttgataatg                                                   20


<210>  13
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  13
cagtgggaga cctcgagaag                                                   20


<210>  14
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  14
tccctcggaa catcagaaac                                                   20


<210>  15
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  15
gagaactttg ccgttgaagc                                                   20


<210>  16
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  16
gcttcctgta ggtggcaatc                                                   20


<210>  17
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  17
tgggaaggca gatgtatctt tcg                                               23


<210>  18
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  18
tgttgactga aggtaggtct ga                                                22


<210>  19
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  19
aaccattaag gtgtcgtatg ctc                                               23


<210>  20
<211>  19
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  20
cgcccaaacc gagagaaca                                                    19


<210>  21
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  21
catccagcta atgtcatgtc tgt                                               23


<210>  22
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  22
ctctggtcac gggatagaat ttc                                               23


<210>  23
<211>  19
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  23
acgcaagctc tgccttttc                                                    19


<210>  24
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  24
cgtgaggact gaagtaccat aga                                               23


<210>  25
<211>  19
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  25
gcgaagccga aaaaggcag                                                    19


<210>  26
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  26
tccgcaggta agtcttcttt agt                                               23


<210>  27
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  27
atggtgacac ccagaccgat                                                   20


<210>  28
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  28
gagaagccat aattggcctg at                                                22


<210>  29
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  29
tcccaaagat ctgccttcac                                                   20


<210>  30
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  30
ttctgcattg tgctgagagg                                                   20


<210>  31
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  31
tcttcttttg aggccaggaa                                                   20


<210>  32
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  32
ggaaagacca agaaaagccc                                                   20


<210>  33
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  33
agttcggtgc tcgaatgata ac                                                22


<210>  34
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  34
aatacgacct tgtgatggaa cg                                                22


<210>  35
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  35
tgaatctcag ccagtggtct t                                                 21


<210>  36
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  36
tcatcacttc ctacggcgat                                                   20


<210>  37
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construction

<400>  37
ttccttttct ccgactctcc tt                                                22


<210>  38
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  38
ccccaagtac caagtgcatg t                                                 21


<210>  39
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  39
tgccagccac ttactgtgaa a                                                 21


<210>  40
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  40
gcctcaccaa caatacccca ta                                                22


<210>  41
<211>  23
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  41
agattggaca acctatggac tga                                               23


<210>  42
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  42
gcactctgtc gaactgaagt ta                                                22


<210>  43
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  43
gaggaggcgt ctccctattc                                                   20


<210>  44
<211>  21
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  44
gcatctggtt gcccctaaaa a                                                 21


<210>  45
<211>  22
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  45
cctgtggtct ttttgaacag ag                                                22


<210>  46
<211>  20
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  46
caactggagg ccctgtatgt                                                   20


<210>  47
<211>  26
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  47
acacacacat aaacagatca tctcgg                                            26


<210>  48
<211>  25
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Synthetic Construct

<400>  48
agtctctgaa cctgtcctgg ttctg                                             25


