                         SEQUENCE LISTING

<110>  Lloyd, R. Stephen
       McCullough, Amanda K.
       Donley, Nathan
 
<120>  SMALL MOLECULE INHIBITORS OF 8-OXOGUANINE DNA GLYCOSYLASE-1 
       (OGG1)

<130>  2140-2

<160>  7     

<170>  PatentIn version 3.5

<210>  1
<211>  17
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  Oligonucleotide


<220>
<221>  misc_feature
<222>  (6)..(6)
<223>  n is a, c, g, or t

<400>  1
tcaccntcgt acgactc                                                      17


<210>  2
<211>  17
<212>  DNA
<213>  Artificial Sequence

<220>
<223>  oligonucleotide

<400>  2
agtggcagca tgctgag                                                      17


<210>  3
<211>  190
<212>  PRT
<213>  Homo sapiens

<400>  3

Gln Asp Pro Ile Glu Cys Leu Phe Ser Phe Ile Cys Ser Ser Asn Asn 
1               5                   10                  15      


Asn Ile Ala Arg Ile Thr Gly Met Val Glu Arg Leu Cys Gln Ala Phe 
            20                  25                  30          


Gly Pro Arg Leu Ile Gln Leu Asp Asp Val Thr Tyr His Gly Phe Pro 
        35                  40                  45              


Ser Leu Gln Ala Leu Ala Gly Pro Glu Val Glu Ala His Leu Arg Lys 
    50                  55                  60                  


Leu Gly Leu Gly Tyr Arg Ala Arg Tyr Val Ser Ala Ser Ala Arg Ala 
65                  70                  75                  80  


Ile Leu Glu Glu Gln Gly Gly Leu Ala Trp Leu Gln Gln Leu Arg Glu 
                85                  90                  95      


Ser Ser Tyr Glu Glu Ala His Lys Ala Leu Cys Ile Leu Pro Gly Val 
            100                 105                 110         


Gly Thr Lys Val Ala Asp Cys Ile Cys Leu Met Ala Leu Asp Lys Pro 
        115                 120                 125             


Gln Ala Val Pro Val Asp Val His Met Trp His Ile Ala Gln Arg Asp 
    130                 135                 140                 


Tyr Ser Trp His Pro Thr Thr Ser Gln Ala Lys Gly Pro Ser Pro Gln 
145                 150                 155                 160 


Thr Asn Lys Glu Leu Gly Asn Phe Phe Arg Ser Leu Trp Gly Pro Tyr 
                165                 170                 175     


Ala Gly Trp Ala Gln Ala Val Ser Val Pro Arg Cys Pro Pro 
            180                 185                 190 


<210>  4
<211>  241
<212>  PRT
<213>  Homo sapiens

<400>  4

Lys Ser Gln Ala Ser Arg Pro Thr Pro Asp Glu Leu Glu Ala Val Arg 
1               5                   10                  15      


Lys Tyr Phe Gln Leu Asp Val Thr Leu Ala Gln Leu Tyr His His Trp 
            20                  25                  30          


Gly Ser Val Asp Ser His Phe Gln Glu Val Ala Gln Lys Phe Gln Gly 
        35                  40                  45              


Val Arg Leu Leu Arg Gln Asp Pro Ile Glu Cys Leu Phe Ser Phe Ile 
    50                  55                  60                  


Cys Ser Ser Asn Asn Asn Ile Ala Arg Ile Thr Gly Met Val Glu Arg 
65                  70                  75                  80  


Leu Cys Gln Ala Phe Gly Pro Arg Leu Ile Gln Leu Asp Asp Val Thr 
                85                  90                  95      


Tyr His Gly Phe Pro Ser Leu Gln Ala Leu Ala Gly Pro Glu Val Glu 
            100                 105                 110         


Ala His Leu Arg Lys Leu Gly Leu Gly Tyr Arg Ala Arg Tyr Val Ser 
        115                 120                 125             


Ala Ser Ala Arg Ala Ile Leu Glu Glu Gln Gly Gly Leu Ala Trp Leu 
    130                 135                 140                 


Gln Gln Leu Arg Glu Ser Ser Tyr Glu Glu Ala His Lys Ala Leu Cys 
145                 150                 155                 160 


Ile Leu Pro Gly Val Gly Thr Lys Val Ala Asp Cys Ile Cys Leu Met 
                165                 170                 175     


Ala Leu Asp Lys Pro Gln Ala Val Pro Val Asp Val His Met Trp His 
            180                 185                 190         


Ile Ala Gln Arg Asp Tyr Ser Trp His Pro Thr Thr Ser Gln Ala Lys 
        195                 200                 205             


Gly Pro Ser Pro Gln Thr Asn Lys Glu Leu Gly Asn Phe Phe Arg Ser 
    210                 215                 220                 


Leu Trp Gly Pro Tyr Ala Gly Trp Ala Gln Ala Ala Gly Ser Asp Ala 
225                 230                 235                 240 


Ser 
    


<210>  5
<211>  275
<212>  PRT
<213>  Homo sapiens

<400>  5

Lys Ser Gln Ala Ser Arg Pro Thr Pro Asp Glu Leu Glu Ala Val Arg 
1               5                   10                  15      


Lys Tyr Phe Gln Leu Asp Val Thr Leu Ala Gln Leu Tyr His His Trp 
            20                  25                  30          


Gly Ser Val Asp Ser His Phe Gln Glu Val Ala Gln Lys Phe Gln Gly 
        35                  40                  45              


Val Arg Leu Leu Arg Gln Asp Pro Ile Glu Cys Leu Phe Ser Phe Ile 
    50                  55                  60                  


Cys Ser Ser Asn Asn Asn Ile Ala Arg Ile Thr Gly Met Val Glu Arg 
65                  70                  75                  80  


Leu Cys Gln Ala Phe Gly Pro Arg Leu Ile Gln Leu Asp Asp Val Thr 
                85                  90                  95      


Tyr His Gly Phe Pro Ser Leu Gln Ala Leu Ala Gly Pro Glu Val Glu 
            100                 105                 110         


Ala His Leu Arg Lys Leu Gly Leu Gly Tyr Arg Ala Arg Tyr Val Ser 
        115                 120                 125             


Ala Ser Ala Arg Ala Ile Leu Glu Glu Gln Gly Gly Leu Ala Trp Leu 
    130                 135                 140                 


Gln Gln Leu Arg Glu Ser Ser Tyr Glu Glu Ala His Lys Ala Leu Cys 
145                 150                 155                 160 


Ile Leu Pro Gly Val Gly Thr Lys Val Ala Asp Cys Ile Cys Leu Met 
                165                 170                 175     


Ala Leu Asp Lys Pro Gln Ala Val Pro Val Asp Val His Met Trp His 
            180                 185                 190         


Ile Ala Gln Arg Asp Tyr Ser Trp His Pro Thr Thr Ser Gln Ala Lys 
        195                 200                 205             


Gly Pro Ser Pro Gln Thr Asn Lys Glu Leu Gly Asn Phe Phe Arg Ser 
    210                 215                 220                 


Leu Trp Gly Pro Tyr Ala Gly Trp Ala Gln Ala Leu Cys Gln Val Ile 
225                 230                 235                 240 


Thr Thr Phe Met Thr Phe Leu Gly Pro His Arg Leu Asp Gln Met Pro 
                245                 250                 255     


Pro Glu Glu Leu Gln Thr Ser Ser Ser Arg Leu Gly Gly Pro Pro Trp 
            260                 265                 270         


Gln Cys Ile 
        275 


<210>  6
<211>  100
<212>  PRT
<213>  Homo sapiens

<400>  6

Val Arg Lys Tyr Phe Gln Leu Asp Val Thr Leu Ala Gln Leu Tyr His 
1               5                   10                  15      


His Trp Gly Ser Val Asp Ser His Phe Gln Glu Val Ala Gln Lys Phe 
            20                  25                  30          


Gln Gly Val Arg Leu Leu Arg Gln Asp Pro Ile Glu Cys Leu Phe Ser 
        35                  40                  45              


Phe Ile Cys Ser Ser Asn Asn Asn Ile Ala Arg Ile Thr Gly Met Val 
    50                  55                  60                  


Glu Arg Leu Cys Gln Ala Phe Gly Pro Arg Leu Ile Gln Leu Asp Asp 
65                  70                  75                  80  


Val Thr Tyr His Gly Phe Pro Ser Leu Gln Ala Leu Ala Gly Pro Pro 
                85                  90                  95      


Trp Gln Cys Ile 
            100 


<210>  7
<211>  255
<212>  PRT
<213>  Homo sapiens

<400>  7

Val Arg Lys Tyr Phe Gln Leu Asp Val Thr Leu Ala Gln Leu Tyr His 
1               5                   10                  15      


His Trp Gly Ser Val Asp Ser His Phe Gln Glu Val Ala Gln Lys Phe 
            20                  25                  30          


Gln Gly Val Arg Leu Leu Arg Gln Asp Pro Ile Glu Cys Leu Phe Ser 
        35                  40                  45              


Phe Ile Cys Ser Ser Asn Asn Asn Ile Ala Arg Ile Thr Gly Met Val 
    50                  55                  60                  


Glu Arg Leu Cys Gln Ala Phe Gly Pro Arg Leu Ile Gln Leu Asp Asp 
65                  70                  75                  80  


Val Thr Tyr His Gly Phe Pro Ser Leu Gln Ala Leu Ala Gly Pro Glu 
                85                  90                  95      


Val Glu Ala His Leu Arg Lys Leu Gly Leu Gly Tyr Arg Ala Arg Tyr 
            100                 105                 110         


Val Ser Ala Ser Ala Arg Ala Ile Leu Glu Glu Gln Gly Gly Leu Ala 
        115                 120                 125             


Trp Leu Gln Gln Leu Arg Glu Ser Ser Tyr Glu Glu Ala His Lys Ala 
    130                 135                 140                 


Leu Cys Ile Leu Pro Gly Val Gly Thr Lys Gly Leu Leu Gly Asn Ala 
145                 150                 155                 160 


Phe Asp Gly His Gln Leu Leu Arg Pro Leu Ile Phe Cys Gln Asp His 
                165                 170                 175     


Leu Arg Glu Gly Pro Pro Ile Gly Arg Gly Asp Ser Gln Gly Glu Glu 
            180                 185                 190         


Leu Glu Pro Gln Leu Pro Ser Ser Leu Ser Ser Ile Pro Tyr Gly Phe 
        195                 200                 205             


Cys Asp His Cys Trp Thr Lys Asp Val Asp Asp Pro Pro Leu Val Thr 
    210                 215                 220                 


His Pro Ser Pro Gly Ser Arg Asp Gly His Met Thr Gln Ala Trp Pro 
225                 230                 235                 240 


Val Lys Val Val Ser Pro Leu Ala Thr Val Ile Gly His Val Met 
                245                 250                 255 


